ʻO ka ʻāpana Corydalis Tetrahydropalmatine (dl-THP)
ʻO Tetrahydropalmatine (THP), i ʻike ʻia hoʻi ʻo dl-THP, Corydalin hydrochloride, a i ʻole Corydalin Tube Extract, he hui i hoʻokaʻawale ʻia he alkaloid isoquinoline. Ua unuhi ʻia mai ka ʻōpū o ka lau nahele Kina ʻo Corydalis yanhusuo. He mea kala ʻole a melemele paha ka THP me kahi ʻono ʻawaʻawa iki a me kahi kiko heheʻe o 147-149°C. He mea hoʻoheheʻe ʻole ia i ka wai akā hoʻoheheʻe nui ʻia i ka ether, chloroform, a me ka ethanol. Hiki ke hoʻoheheʻe ʻia kona paʻakai hydrochloride a me sulfate i ka wai.
Ua aʻo ʻia ʻo THP no nā hopena pharmacological like ʻole, me kona analgesic, anesthetic, neuroprotective, antiplatelet aggregation, antiulcer, antitumor, a me nā waiwai anti-addiction. Ua manaʻoʻiʻo ʻia e hoʻohana i kona mau hopena analgesic ma ka hoʻololi ʻana i ka hana receptor dopamine waena a ua hōʻike i ka hiki ke pale i nā neurons mai ka hōʻeha ischemic. Eia kekahi, ua hōʻike ʻo THP i nā hopena antiplatelet aggregation a ua noiʻi ʻia no kona hiki ke mālama i nā ʻōpū, ka pale ʻana i ka ulu ʻana o nā cell tumor, a me ke kōkua ʻana i ka hoʻohui lāʻau.
Ma keʻano holoʻokoʻa, ʻo Tetrahydropalmatine (dl-THP) kahi hui me nā ʻano pharmacological like ʻole a ua lilo ia i kumuhana o ka noiʻi nui no kāna mau noi therapeutic hiki. No ka ʻike hou aku e hoʻokaʻaʻikegrace@biowaycn.com.
Eia nā hiʻohiʻona huahana o Tetrahydropalmatine (THP) me ko lākou mau pono olakino:
1. Nā Waiwai Analgesic:Hōʻike ʻo THP i nā hopena analgesic ma ka hoʻololi ʻana i ka hana o ka mea loaʻa dopamine waena, e hāʻawi ana i ka hōʻoluʻolu ʻeha me ka ʻole o ka hiki ke hoʻopili nui.
2. Nā hopena palekana neuro:Ua hōʻike ʻo THP i ka hiki ke pale i nā neurons mai ka hōʻeha ischemic, e hōʻemi ana i ka apoptosis neuronal, a me ka hoʻohaʻahaʻa ʻana i nā pae glutamate i loko o ka lolo, kahi e hiki ai ke kōkua i kāna mau waiwai neuroprotective.
3. Hoʻohuihui Antiplatelet:Ua ʻike ʻia ua kāohi ʻo THP i ka hōʻiliʻili ʻana o ka platelet, e hōʻemi ana i ka pilikia o ke kūkulu ʻia ʻana o ke koko a me nā hanana cardiovascular e pili ana.
4. Kākoʻo Ola Kino:Ua hōʻike ʻo THP i nā hopena anti-ulcer a hiki ke kōkua i ka hōʻemi ʻana i ka hoʻokuʻu ʻana o ka waikawa gastric, e hāʻawi ana i ka hōʻoluʻolu mai nā ʻeha gastric a me nā kūlana pili.
5. Hana Antitumor Hiki:Ua hōʻike ʻo THP i nā hopena cytotoxic ma nā pūnaewele tumor, e hōʻike ana i kahi kuleana kūpono i ke kāohi ʻana i ka ulu ʻana o ka tumor.
6. Nā Waiwai Kū'ē i ka ʻAʻai:Ua aʻo ʻia ʻo THP no kona hiki ke hōʻoluʻolu i nā hōʻailona haʻalele e pili ana i ka opioid a me ka stimulant addiction, e hāʻawi ana i ka ʻōlelo hoʻohiki i ka mālama ʻana i ka ʻona a me ka pale ʻana i ka relapse.
Hōʻike kēia mau hiʻohiʻona i nā pono olakino like ʻole a me nā hoʻohana therapeutic kūpono o Tetrahydropalmatine (THP).
No nā alkaloids isoquinoline ʻo Tetrahydropydalin (dl-THP) a he alkaloid ia, ʻo ia hoʻi ma ka genus Corydalis lucidum (Yan Hu Suo), akā i nā mea kanu ʻē aʻe e like me Stephania rotunda. Loaʻa i kēia mau mea kanu nā hoʻohana kuʻuna i ka lāʻau lapaʻau Kina.He mea kanu mau ka Corydalis, he 10 a 20 cm ke kiʻekiʻe, me nā ʻōpuʻu poepoe. He pōkole a lahilahi kona mau kumu ma luna o ka honua, me kahi unahi ma luna o ke kumu. Ua like ke ʻano o nā lau basal a me nā lau cauline, me nā kumu; ua ʻokoʻa nā lau cauline, me 2 a me 3 mau lau hui. ʻO ka lua o ka lau e māhele pinepine ʻole ʻia a ua lobedi hohonu. He oblong, oval, a oval paha nā lau liʻiliʻi. Linear, ma kahi o 2 cm ka lōʻihi, me ka ʻoki ʻoi a ʻoi paha a me nā lihi maʻemaʻe. He ʻano raceme kona inflorescence, me nā lau terminal a i ʻole nā lau ʻē aʻe; he lanceolate ākea nā bracts; he ʻulaʻula-poni nā pua a ulu pālahalaha ma nā pedicels lahilahi, ma kahi o 6 mm ka lōʻihi; hāʻule mua ka calyx; he 4 nā petals a he 2 nā whorls waho. ʻOi aku ka nui o nā ʻāpana, me nā lihi poni a me ke kikowaena poni-uliuli. Aia kekahi ʻāpana luna, a hoʻolōʻihi ka huelo i loko o kahi spur lōʻihi. ʻO ka lōʻihi o ka spur no ka hapalua o ka lōʻihi holoʻokoʻa. ʻOi aku ka haiki o nā ʻāpana 2 o loko ma mua o nā ʻāpana 2 o waho. He poni uliuli ka ʻaoʻao o luna a ua ho'ōla ʻia, a he poni ka ʻāpana o lalo; ʻEono nā stamens, a ua hoʻopili ʻia nā filaments i ʻelua mau puʻupuʻu, me 3 anthers kēlā me kēia; he palahalaha-cylindrical ka ovary, he pōkole a lahilahi ke ʻano, a ʻelua ka stigma, e like me ka pulelehua liʻiliʻi. He capsule kona hua. Hoʻoulu nui ʻia ʻo Corydalis ma nā mauna a i ʻole nā pāpū mauʻu. ʻO nā wahi hana nui e pili ana iā Zhejiang, Hebei, Shandong, Jiangsu, a me nā wahi ʻē aʻe.
| Ka nānā ʻana | Nā kikoʻī |
| Hoʻāʻo | ʻO Tetrahydropalmatine ≥98% |
| helehelena | Pauka melemele māmā a i keʻokeʻo |
| Lehu | ≤0.5% |
| ka makū | ≤5.0% |
| Nā mea pepehi lāʻau make | Maikaʻi ʻole |
| Nā metala kaumaha | ≤10ppm |
| Pb | ≤2.0ppm |
| As | ≤2.0ppm |
| ʻAla | ʻAno |
| Ka nui o ka ʻāpana | 100% a hiki i ka 80 mesh |
| ʻO ka maʻi mikrobiolo: | |
| Ka huina o nā bacteria | ≤1000cfu/g |
| Nā fungi | ≤100cfu/g |
| ʻO Salmgosella | Maikaʻi ʻole |
| Koli | Maikaʻi ʻole |
Eia nā ʻoihana hoʻopili huahana o Tetrahydropalmatine (THP):
1. Nā lāʻau lapaʻau:Hoʻohana ʻia ʻo THP i ka ʻoihana lāʻau lapaʻau no ka hoʻomohala ʻana i nā lāʻau lapaʻau hoʻokele ʻeha a me nā lāʻau neuroprotective.
2. Nā meaʻai nutraceutical:Hoʻohana ʻia ka THP i ka ʻoihana nutraceutical no ka hana ʻana i nā mea hoʻohui e pili ana i ka hōʻoluʻolu ʻeha a me ke kākoʻo olakino ʻōpū.
3. ʻEnehana Olaola:Loaʻa iā THP nā noi i loko o ka biotechnology no ka noiʻi ʻana i nā hoʻoponopono antiplatelet a me nā mea kōkua lapaʻau kanesa.
4. Mālama Ola:Ua hoʻokomo ʻia ʻo THP i loko o nā huahana mālama ola no ka mālama ʻana i ka ʻona a me nā hōʻailona haʻalele e pili ana i ka hoʻohana ʻana i ka opioid a me ka stimulant.
5. Nā mea hoʻonaninani:Ua ʻimi ʻia ʻo THP i loko o nā cosmeceuticals no ke olakino ʻili a me nā noi anti-inflammatory.
Hōʻike kēia mau ʻoihana i nā hoʻohana like ʻole o Tetrahydropalmatine (THP) i nā ʻano hoʻomohala huahana a me nā noiʻi like ʻole.
Hana ʻia kā mākou huahana me ka hoʻohana ʻana i nā ana hoʻomalu maikaʻi koʻikoʻi a pili i nā kūlana kiʻekiʻe o nā kaʻina hana. Hoʻoikaika mākou i ka palekana a me ka maikaʻi o kā mākou huahana, e hōʻoia ana e hoʻokō ia i nā koi hoʻoponopono a me nā palapala hōʻoia o ka ʻoihana. ʻO kēia kūpaʻa i ka maikaʻi e manaʻo e hoʻokumu i ka hilinaʻi a me ka hilinaʻi i ka hilinaʻi o kā mākou huahana. Penei ke kaʻina hana maʻamau:
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