ʻO Stephania Extract Cepharanthine Powder

Inoa Huahana: Stephania Japonica Extract
Kumu Latina: Stephania cephalantha Hayata (Stephania japonica (Thunb.)Miers) / Stephania epigaea Lo / Stephania yunnanensis HSLo.
ʻAno: Keʻokeʻo, hina hina keʻokeʻo pauka
Mea Hana: Cepharanthine 80%-99% HPLC
ʻĀpana i hoʻohana ʻia: Tuber/Root
Noi: Nā huahana mālama ola kino
Kiko heheʻe: 145-155°
Hoʻohuli kikoʻī: D20+277°(c=2inchloroform)
Kikowaena paila: 654.03°C (manaʻo maʻamau)
Ka nui: 1.1761 (kuhikuhi maʻamau)
ʻIkepili refractive: 1.5300 (kuhikuhi)
Nā kūlana mālama: ke kinoea ma lalo o ka wai (naikokene a i ʻole Argon) ma 2-8°C
Ka hoʻoheheʻe ʻia: Hoʻoheheʻe ʻia i loko o SO (35mg/mL) a i ʻole ethanol (20mg/mL)
Ka helu ʻakika (pKa):7.61 ± 0.20 (Wānana ʻia)


Nā kikoʻī huahana

Nā ʻIke ʻē aʻe

Nā Lepili Huahana

Hoʻolauna Huahana

ʻO ka pauka ʻo Stephania Extract Cepharanthine kahi mea i loaʻa mai nā ʻōpū o ka mea kanu ʻo Stephania cephalantha Hayata (Stephania japonica (Thunb.) Miers) a i ʻole Stephania epigaea Lo/ Stephania yunnanensis HSLo. He huahana kūlohelohe ʻo Cepharanthine i hoʻokaʻawale ʻia mai kēia mea kanu a ua lilo ia i kumuhana o nā haʻawina like ʻole ma muli o kona mau waiwai pharmacological hiki. Ua ʻike ʻia he mau hana anti-SARS-CoV-2, e hōʻike ana i ka pono i ka hoʻopau ʻana i ka hoʻolaha ʻana o ka viral. Eia kekahi, ua hōʻike ʻo Cepharanthine i ka hiki ke hoʻohuli i ke kūʻē ʻana o ka lāʻau lapaʻau P-glycoprotein (P-gp) i kekahi mau cell a hoʻonui i ka ʻike o nā mea anticancer i nā hiʻohiʻona hoʻokolohua. Eia kekahi, ua hōʻike ʻia he mau hopena inhibitory i nā enzymes cytochrome P450 o ke ake kanaka CYP3A4, CYP2E1, a me CYP2C9, a pili pū me nā hopena antitumor, anti-inflammatory, a me antinociceptive.
I ka hōʻuluʻulu manaʻo, ʻo Stephania Extract Cepharanthine Powder kahi ʻano pauka o ka huahana kūlohelohe ʻo Cepharanthine i loaʻa mai ka mea kanu Stephania cephalantha, ka mea i hōʻike i ka hiki ke hana i nā noi pharmacological like ʻole.

Kikoʻī (COA)

Huahana ʻO Cepharanthine
CAS 481-49-2
Hoʻāʻo 80%~99%
helehelena Pauka keʻokeʻo
Hoʻopili ʻana ʻEke 1KG/Foil
Mea Nā kikoʻī
helehelena pauka keʻokeʻo hina, ʻala kūlike, hygroscopic kiʻekiʻe
Ka ʻike ʻana TLC: Hoʻonā maʻamau a me ka hoʻonā hoʻāʻo i kahi like, RF
Hoʻāʻo (Kumu maloʻo) 98.0%--102.0%
ʻIke Optical Kūikawā -2.4°~ -2.8°
PH 4.5~7.0
Nā Metala Kaumaha (Ma ke ʻano he Pb) ≤10ppm
As ≤1ppm
Pb ≤0.5ppm
Cd ≤1ppm
Hg ≤0.1ppm
Mea pili ʻAʻole ʻoi aku ka nui o ka wahi ma mua o ka wahi hoʻonā maʻamau
Mea hoʻoheheʻe koena <0.5%
Ka nui o ka wai <2%

Nā Hiʻohiʻona Huahana

ʻO ka Stephania Extract Cepharanthine Powder kahi huahana kūlohelohe i loaʻa mai ka mea kanu ʻo Stephania cephalantha Hayata. Ua ʻike ʻia he mau waiwai pharmacological kekahi, me:
1. Nā hana kū'ē iā SARS-CoV-2
2. Nā hopena pale i ka hoʻolaha ʻana o ka viral
3. Hoʻohuli ʻia o ke kū'ē ʻana o ka lāʻau lapaʻau i hoʻopili ʻia e P-glycoprotein
4. Hoʻonui i ka ʻike i nā mea anticancer
5. Nā hopena hoʻopaʻa i nā enzyme cytochrome P450 o ke ake kanaka CYP3A4, CYP2E1, a me CYP2C9
6. Nā hopena antitumor, anti-inflammatory, a me antinociceptive

He aha ke ʻano o ka hana ʻana o Cepharanthine?

Hoʻomaka ka biosynthesis o cepharanthine ma Stephania me ka condensation o dopamine a me 4-hydroxyphenylacetaldehyde (4-HPAA, 5) ma o norcoclaurine synthase (NCS), e hua mai ana i ka norcoclaurine.

He aha ka solubility o Cepharanthine?

Hiki ke hoʻoheheʻe ʻia ʻo Cepharanthine i loko o nā mea hoʻoheheʻe organik e like me ka ethanol, DMSO, a me ka dimethyl formamide (DMF). ʻO ka solubility o ka cepharanthine i loko o kēia mau mea hoʻoheheʻe ma kahi o 2, 5, a me 10 mg/ml, kēlā me kēia. He kakaikahi ka hoʻoheheʻe ʻia ʻana o Cepharanthine i loko o nā buffers aqueous.

Nā noi

ʻO nā ʻoihana noi no Stephania Extract Cepharanthine Powder e komo pū me Pharmaceutical, Nutraceutical, Biotechnology, a me Herbal Medicine, ʻo nā noi nui penei:
Ka hiki ke hoʻohana ʻia i nā lāʻau lapaʻau antiviral
Ka hiki ke lilo i mea kōkua i ka mālama ʻana i ka maʻi kanesa
Ka hiki ke hoʻohana ʻia i nā lāʻau anti-inflammatory
Ka hiki ke lilo i mea hoʻōla analgesic
Hōʻike kēia mau noi i nā hoʻohana like ʻole o Stephania Extract Cepharanthine Powder i nā ʻano therapeutic like ʻole.


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